Peptide-Appended Permethylated β-Cyclodextrins with Hydrophilic and Hydrophobic Spacers
نویسندگان
چکیده
منابع مشابه
Peptide-Appended Permethylated β-Cyclodextrins with Hydrophilic and Hydrophobic Spacers
A novel synthetic methodology, employing a combination of the strain-promoted azide-alkyne cycloaddition and maleimide-thiol reactions, for the preparation of permethylated β-cyclodextrin-linker-peptidyl conjugates is reported. Two different bifunctional maleimide cross-linking probes, the polyethylene glycol containing hydrophilic linker bicyclo[6.1.0] nonyne-maleimide and the hydrophobic 5'-d...
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ژورنال
عنوان ژورنال: Bioconjugate Chemistry
سال: 2017
ISSN: 1043-1802,1520-4812
DOI: 10.1021/acs.bioconjchem.7b00319